产品属性:
产品名称 | ABP 688 |
规格 | 10 mg、50 mg |
货号 | EY-01Y14065 |
Cas No.: 924298-51-1
别名: N/A
化学名: N/A
分子式: C15H16N2O
分子量: 240.3
溶解度: DMSO: 100 mM
储存条件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
产品描述:
High affinity human mGlu5 receptor antagonist (Ki = 1.7 nM). Inhibits glutamate-induced calcium release from L(tk-) cells expressing human mGlu5 receptors (IC50 = 2.3 nM).Hintermann et al (2007) ABP688, a novel selective and high affinity ligand for the labeling of mGlu5 receptors: identification, in vitro pharmacology, pharmacokinetic and biodistribution studies. Bioorg.Med.Chem. 15 903 PMID:17110115
特别提醒公司产品仅供科研使用